SCHEMBL5371022

SCHEMBL5371022

O=C(NC(C(=O)CSc1ccccc1)C1CCNCC1)c1ccc(O)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.49
POLB P06746 2/20 0.49
PPARG P37231 1/20 0.49
NCOA2 Q15596 1/20 0.49
NCOA1 Q15788 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
SMYD3 Q9H7B4 3/20 0.39
AKT1 P31749 2/20 0.38
CDK2 P24941 1/20 0.38
USP2 O75604 1/20 0.38
CASP3 P42574 1/20 0.37
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
OPRD1 P41143 1/20 0.36
KDM4E B2RXH2 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CTSL P07711 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362924 0.81 KMT2A (0.41) KMT2APOLBMEN1SMYD3AKT1
SCHEMBL5367918 0.80 ALDH1A1 (0.41) KMT2AMEN1MAPTSMYD3AKT1
SCHEMBL5366087 0.75 HPGD (0.44) KMT2APOLBMEN1MAPTSMYD3
SCHEMBL5370964 0.74 KMT2A (0.46) KMT2APOLBPPARGNCOA2NCOA1
SCHEMBL5371067 0.74 NPC1 (0.42) SMYD3AKT1CDK2NPC1RAB9A
SCHEMBL5364811 0.73 MEN1 (0.42) KMT2AMEN1SMYD3AKT1CDK2
SCHEMBL5370713 0.72 CTSL (0.42) KMT2AMEN1SMYD3CTSL
SCHEMBL5362898 0.72 SMYD3 (0.43) KMT2AMEN1MAPTSMYD3NPC1
SCHEMBL5366736 0.72 AKT1 (0.42) SMYD3AKT1NPC1RAB9A
SCHEMBL5360331 0.71 SCN3A (0.39) SMYD3AKT1CDK2OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed