SCHEMBL5366324

SCHEMBL5366324

Cc1c(Br)ccc2c1C(=Cc1ccc(F)cc1C(F)(F)F)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
FLT3 P36888 5/20 0.42
MDM2 Q00987 3/20 0.38
ADORA2A P29274 1/20 0.38
ALK Q9UM73 1/20 0.37
TGM2 P21980 1/20 0.37
PDGFRB P09619 1/20 0.36
RPS6KA3 P51812 1/20 0.36
KDR P35968 1/20 0.35
NTRK1 P04629 1/20 0.35
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7134441 0.85 MYC (0.43) MEN1KMT2AFLT3ADORA2AKDR
SCHEMBL7136928 0.84 KMT2A (0.37) MEN1KMT2AFLT3MDM2ADORA2A
SCHEMBL5362861 0.84 MEN1 (0.46) MEN1KMT2AFLT3MDM2ALK
SCHEMBL7138200 0.84 MEN1 (0.47) MEN1KMT2AFLT3MDM2ALK
SCHEMBL5357855 0.82 MEN1 (0.39) MEN1KMT2AFLT3KDRCCNE1
SCHEMBL5368774 0.80 MEN1 (0.37) MEN1KMT2AFLT3MDM2ALK
SCHEMBL5366373 0.78 KDR (0.36) MEN1KMT2AFLT3PDGFRBKDR
SCHEMBL7139913 0.77 RAF1 (0.42) MEN1KMT2APDGFRBNTRK1
SCHEMBL7136994 0.77 MAOA (0.44) MEN1KMT2AFLT3PDGFRBKDR
SCHEMBL7138309 0.76 MEN1 (0.51) MEN1KMT2AFLT3MDM2PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK MEN1 3855/4885KMT2A 4060/4885FLT3 395/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.