SCHEMBL5366486

SCHEMBL5366486

CS(=O)(=O)Nc1ccc(C(=O)NCC2CN(C(=O)OCc3ccccc3)CCO2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.56
TSHR P16473 1/20 0.56
ADRB1 P08588 5/20 0.49
ENPP2 Q13822 2/20 0.45
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
GAA P10253 2/20 0.42
F2 P00734 1/20 0.42
PLG P00747 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
TPSAB1 Q15661 1/20 0.42
TPSD1 Q9BZJ3 1/20 0.42
TPSG1 Q9NRR2 1/20 0.42
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425338 1.00 SMN1; SMN2 (0.56) SMN1; SMN2TSHRADRB1ENPP2ALDH1A1
SCHEMBL14425436 0.87 MEN1 (0.50) SMN1; SMN2ENPP2ALDH1A1MEN1KMT2A
SCHEMBL5368740 0.87 MEN1 (0.50) SMN1; SMN2ENPP2ALDH1A1MEN1KMT2A
SCHEMBL14425317 0.87 MEN1 (0.50) SMN1; SMN2ENPP2ALDH1A1MEN1KMT2A
SCHEMBL5367296 0.83 GRIN2B (0.51) SMN1; SMN2ENPP2MEN1KMT2ANPSR1
SCHEMBL5362334 0.83 ENPP2 (0.47) SMN1; SMN2ENPP2ALDH1A1KDM4EMEN1
SCHEMBL5369961 0.83 MEN1 (0.46) ENPP2MEN1KMT2ANPSR1GAA
SCHEMBL5364470 0.83 TPSAB1 (0.62) SMN1; SMN2ADRB1ALDH1A1KDM4EF2
SCHEMBL5374908 0.82 ENPP2 (0.48) SMN1; SMN2ENPP2MEN1KMT2ANPSR1
SCHEMBL14425340 0.82 ENPP2 (0.48) SMN1; SMN2ENPP2MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed