SCHEMBL5367040

SCHEMBL5367040

CCCCCCCc1ccc2ccccc2n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.61
GPBAR1 Q8TDU6 4/20 0.55
TLR8 Q9NR97 1/20 0.51
CYSLTR1 Q9Y271 3/20 0.51
CYSLTR2 Q9NS75 2/20 0.51
PDE10A Q9Y233 1/20 0.49
LTB4R Q15722 1/20 0.47
MAPK1 P28482 2/20 0.46
CYP1A2 P05177 2/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
CYP2C19 P33261 1/20 0.46
HIF1A Q16665 1/20 0.46
MEN1 O00255 1/20 0.46
GMNN O75496 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28561362 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL797638 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL28545037 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL6114801 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL6115276 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL29903853 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL6114960 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL2514450 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL6115301 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2
SCHEMBL29369286 1.00 KCNH2 (0.61) KCNH2GPBAR1TLR8CYSLTR1CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180057852-A1 Spectrometric Analysis of Microbes MICROMASS UK LIMITED (GB) 2018-03-01 US disclosed
CN-107667288-A Spectral analysis of microorganisms 英国质谱公司 2018-02-06 CN disclosed
CN-104211620-B The autofrettage of bi-quaternary ammonium salt and its intermediate Wako-chem Industries Co., Ltd. (JP) 2016-05-25 CN disclosed
EP-2821395-A2 Novel disulfonic acid ester as an additive for an electrolyte for a lithium secondary battery Wako Pure Chemical Industries, Ltd. (JP) 2015-01-07 EP disclosed
CN-104211620-A PROCESS FOR PRODUCTION OF BIS-QUATERNARY AMMONIUM SALT, AND NOVEL INTERMEDIATE WAKO PURE CHEM IND LTD 2014-12-17 CN disclosed
US-8716513-B2 Process for production of bis-quaternary ammonium salt, and novel intermediate WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2014-05-06 US disclosed
EP-2463266-A1 PROCESS FOR PRODUCTION OF BIS-QUATERNARY AMMONIUM SALT, AND NOVEL INTERMEDIATE Wako Pure Chemical Industries, Ltd. (JP) 2012-06-13 EP disclosed
CN-102482197-A Process for producing diquaternary ammonium salt and novel intermediate WAKO PURE CHEM IND LTD 2012-05-30 CN disclosed
US-20120130107-A1 PROCESS FOR PRODUCTION OF BIS-QUATERNARY AMMONIUM SALT, AND NOVEL INTERMEDIATE WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 2012-05-24 US disclosed
WO-2007008769-A2 USE OF PSEUDAN AND PSEUDAN INCLUSION BODIES GEORGE MASON UNIVERSITY (US) 2007-01-18 WO disclosed
WO-2005069989-A2 METHODS FOR IDENTIFYING CANDIDATE COMPOUNDS FOR TREATING, REDUCING, OR PREVENTING PATHOGENIC INFECTIONS THE GENERAL HOSPITAL CORPORATION (US) 2005-08-04 WO disclosed
EP-0529452-B1 1,7-Condensed 3-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them SOLVAY PHARM GMBH (DE) 1998-11-11 EP disclosed
US-5324725-A Antiinflammatory agent, antiallergen KALI-CHEMIE PHARMA GMBH (DE) 1994-06-28 US disclosed
CN-1069732-A 1, the 2-that 7-a pair of horses going side by side is closed (piperazine alkyl) indole derivatives and preparation method and intermediate product and the medicament that contains these compounds KALI CHEMIE PHARMA GMBH (DE) 1993-03-10 CN disclosed
EP-0529452-A2 1,7-Condensed 2-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them Kali-Chemie Pharma GmbH (DE) 1993-03-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120130107-A1 PROCESS FOR PRODUCTION OF BIS-QUATERNARY AMMONIUM SALT, AND NOVEL INTERMEDIATE ASS1, C1S, FHIT KCNH2 288/4885GPBAR1 1447/4885TLR8 3836/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.