SCHEMBL5367070

SCHEMBL5367070

Cc1ccc(Cc2n[nH]c(=O)cc2C)cc1Oc1cccc(Cl)n1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
SLC22A12 Q96S37 1/20 0.35
PARP1 P09874 12/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
PTGS2 P35354 1/20 0.34
ADORA2A P29274 1/20 0.33
GRM4 Q14833 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CCNE2 O96020 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14570951 0.85 CYP3A4 (0.36) CYP3A4CYP2C9TSHRCYP2C19SLC22A12
SCHEMBL5365237 0.81 CYP3A4 (0.36) CYP3A4CYP2C9TSHRCYP2C19SLC22A12
SCHEMBL5373462 0.75 CYP3A4 (0.41) CYP3A4CYP2C9TSHRCYP2C19PARP1
SCHEMBL5364878 0.73 PARP1 (0.43) CYP3A4CYP2C9TSHRCYP2C19PARP1
SCHEMBL5377601 0.73 PARP1 (0.38) CYP3A4CYP2C9TSHRCYP2C19PARP1
SCHEMBL5368822 0.72 PARP1 (0.33) CYP3A4CYP2C9TSHRCYP2C19PARP1
SCHEMBL5364936 0.71 PRMT5 (0.40) CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5370838 0.69 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19
SCHEMBL14570722 0.67 CYP3A4 (0.34) CYP3A4CYP2C9TSHRCYP2C19SLC22A12
SCHEMBL5368939 0.67 CYP3A4 (0.64) CYP3A4CYP2C9TSHRCYP2C19PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed