SCHEMBL5367220

SCHEMBL5367220

O=c1ccc(Cc2cc(Cc3cc(Cl)cc(Cl)c3)c3occc3c2)n[nH]1

nearest known ligand 0.84

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.84
AKR1B1 P15121 1/20 0.33
KMT2A Q03164 1/20 0.31
THRA P10827 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370940 0.87 CYP3A4 (0.78) CYP3A4AKR1B1KMT2ATHRATHRB
SCHEMBL5373808 0.85 CYP3A4 (0.69) CYP3A4AKR1B1THRATHRB
SCHEMBL5372498 0.83 CYP3A4 (0.83) CYP3A4AKR1B1THRATHRB
SCHEMBL5368912 0.83 CYP3A4 (0.83) CYP3A4AKR1B1THRATHRB
SCHEMBL5374414 0.81 CYP3A4 (0.67) CYP3A4AKR1B1
SCHEMBL5368824 0.81 CYP3A4 (0.70) CYP3A4AKR1B1
SCHEMBL5370463 0.79 CYP3A4 (0.63) CYP3A4
SCHEMBL5377164 0.78 CYP3A4 (0.80) CYP3A4AKR1B1THRATHRB
SCHEMBL5368514 0.78 CYP3A4 (0.80) CYP3A4KMT2ATHRATHRB
SCHEMBL5385893 0.77 CYP3A4 (0.58) CYP3A4AKR1B1KMT2ATHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed