SCHEMBL5370463

SCHEMBL5370463

COc1ccccc1Cc1cc(Cc2ccc(=O)[nH]n2)cc2ccoc12

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.63
CNR2 P34972 9/20 0.40
GPR55 Q9Y2T6 4/20 0.40
GPR18 Q14330 1/20 0.40
AR P10275 1/20 0.39
CNR1 P21554 2/20 0.38
KDM1A O60341 1/20 0.35
GAA P10253 1/20 0.35
HSD17B10 Q99714 1/20 0.35
RCOR1 Q9UKL0 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374414 0.85 CYP3A4 (0.67) CYP3A4AR
SCHEMBL5370940 0.84 CYP3A4 (0.78) CYP3A4CNR2GPR55
SCHEMBL5367220 0.79 CYP3A4 (0.84) CYP3A4
SCHEMBL7276901 0.79 AR (0.55) CNR2GPR55ARKDM1AGAA
SCHEMBL5368824 0.78 CYP3A4 (0.70) CYP3A4AR
SCHEMBL5373808 0.78 CYP3A4 (0.69) CYP3A4
SCHEMBL5370307 0.77 CYP3A4 (0.80) CYP3A4
SCHEMBL5385611 0.75 CYP3A4 (0.62) CYP3A4
SCHEMBL5376979 0.74 CYP3A4 (0.61) CYP3A4CNR2
SCHEMBL5372604 0.73 CYP3A4 (0.71) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed