SCHEMBL5370940

SCHEMBL5370940

O=c1ccc(Cc2cc(Cc3ccccc3)c3occc3c2)n[nH]1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.78
POLB P06746 1/20 0.36
AKR1B1 P15121 1/20 0.35
CYP1A2 P05177 1/20 0.35
CTRC Q99895 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GPR55 Q9Y2T6 2/20 0.33
MPO P05164 1/20 0.33
TPO P07202 1/20 0.33
EPX P11678 1/20 0.33
MEN1 O00255 1/20 0.33
ELANE P08246 1/20 0.33
KMT2A Q03164 1/20 0.33
CNR2 P34972 1/20 0.33
CFD P00746 1/20 0.33
THRA P10827 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373808 0.89 CYP3A4 (0.69) CYP3A4AKR1B1THRATHRB
SCHEMBL5367220 0.87 CYP3A4 (0.84) CYP3A4AKR1B1KMT2ATHRATHRB
SCHEMBL5374414 0.87 CYP3A4 (0.67) CYP3A4AKR1B1ALDH1A1MPOCFD
SCHEMBL5368824 0.84 CYP3A4 (0.70) CYP3A4AKR1B1MPO
SCHEMBL5370463 0.84 CYP3A4 (0.63) CYP3A4GPR55CNR2
SCHEMBL5370307 0.81 CYP3A4 (0.80) CYP3A4AKR1B1CYP1A2MEN1KMT2A
SCHEMBL5373725 0.81 CYP3A4 (0.80) CYP3A4POLBCYP1A2ALDH1A1SMN1; SMN2
SCHEMBL5351260 0.78 AKR1B1 (0.51) CYP3A4POLBAKR1B1CYP1A2ALDH1A1
SCHEMBL5368780 0.76 CYP3A4 (0.74) CYP3A4POLBAKR1B1CYP1A2ALDH1A1
SCHEMBL5365374 0.76 CYP3A4 (0.68) CYP3A4AKR1B1ALDH1A1RAB9ATHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed