SCHEMBL5367265

SCHEMBL5367265

COc1ccc2ncn(CC(=O)NCCN(C)C3CCCCC3)c2c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.52
MTNR1B P49286 3/20 0.52
MAPT P10636 4/20 0.42
TP53 P04637 3/20 0.42
ATM Q13315 6/20 0.42
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CDYL2 Q8N8U2 1/20 0.40
CDYL Q9Y232 1/20 0.40
CDY1; CDY1B Q9Y6F8 1/20 0.40
PDE2A O00408 3/20 0.39
PDE3B Q13370 3/20 0.39
PDE3A Q14432 3/20 0.39
P2RY12 Q9H244 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3606205 0.93 TP53 (0.45) MTNR1AMTNR1BMAPTTP53ATM
SCHEMBL5345349 0.88 TRPA1 (0.43) MAPTTP53ATMALDH1A1L3MBTL1
SCHEMBL13115367 0.87 TRPA1 (0.42) MAPTTP53ATMALDH1A1L3MBTL1
SCHEMBL13115590 0.84 ATM (0.47) ATM
SCHEMBL5367271 0.83 MTNR1A (0.53) MTNR1AMTNR1BTP53ALDH1A1CDYL2
SCHEMBL3605821 0.83 CCNE1 (0.43) MAPTTP53ATML3MBTL1
SCHEMBL3602186 0.82 TP53 (0.41) MAPTTP53ALDH1A1P2RY12
SCHEMBL3597098 0.81 KMT2A (0.42) MAPTTP53ALDH1A1L3MBTL1
SCHEMBL3599700 0.79 ATM (0.42) MAPTTP53ATMALDH1A1
SCHEMBL13115365 0.77 TRPV1 (0.46) MAPTTP53ATMALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
WO-2007115231-A2 CXCR4 MODULATORS CHEMOCENTRYX, INC. (US) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275965-A1 CXCR4 modulators CXCL12, CXCR4, CXCR1 MTNR1A 1079/4885MTNR1B 833/4885MAPT 2809/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.