SCHEMBL5367904

SCHEMBL5367904

O=C(NCC1CCN(C(=O)COc2ccccc2)CC1)c1ccc(O)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ME2 P23368 1/20 0.56
ME1 P48163 1/20 0.56
ME3 Q16798 1/20 0.56
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
KDM4E B2RXH2 2/20 0.54
PKM P14618 1/20 0.54
ALDH1A1 P00352 3/20 0.51
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
CHRM4 P08173 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366718 0.89 SMN1; SMN2 (0.56) MEN1KMT2AKDM4EPKMALDH1A1
SCHEMBL5370693 0.89 KMT2A (0.57) MEN1KMT2AKDM4EPKMALDH1A1
SCHEMBL5362882 0.89 MMP13 (0.56) KMT2AKDM4EPKMALDH1A1POLB
SCHEMBL5370951 0.89 HPGD (0.57) MEN1KMT2AKDM4EPKMALDH1A1
SCHEMBL5366075 0.85 MEN1 (0.56) MEN1KMT2AKDM4EPKMALDH1A1
SCHEMBL5521812 0.81 HDAC3 (0.51) MEN1KMT2ACHRM4HDAC3HDAC4
SCHEMBL5523321 0.81 HDAC3 (0.51) MEN1KMT2ACHRM4HDAC3HDAC4
SCHEMBL5521806 0.81 HDAC3 (0.51) MEN1KMT2ACHRM4HDAC3HDAC4
SCHEMBL5362915 0.81 HDAC6 (0.60) ME2ME1ME3KDM4EPKM
SCHEMBL6536256 0.81 KDM4E (0.55) MEN1KMT2AKDM4EPKMCHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed