SCHEMBL5362882

SCHEMBL5362882

Cc1ccc(OCC(=O)N2CCC(CNC(=O)c3ccc(O)cc3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.56
ALDH1A1 P00352 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
KMT2A Q03164 1/20 0.53
POLB P06746 1/20 0.49
HTT P42858 1/20 0.49
USP2 O75604 1/20 0.48
HPGD P15428 1/20 0.48
FKBP1A P62942 1/20 0.48
TP53 P04637 2/20 0.47
KDM4E B2RXH2 2/20 0.47
PKM P14618 2/20 0.47
ADRB2 P07550 1/20 0.46
F2 P00734 1/20 0.46
PLG P00747 1/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
TPSAB1 Q15661 1/20 0.46
TPSD1 Q9BZJ3 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370693 0.89 KMT2A (0.57) ALDH1A1SMN1; SMN2KMT2APOLBFKBP1A
SCHEMBL5366718 0.89 SMN1; SMN2 (0.56) ALDH1A1SMN1; SMN2KMT2APOLBHTT
SCHEMBL5367904 0.89 ME2 (0.56) ALDH1A1SMN1; SMN2KMT2APOLBUSP2
SCHEMBL5370951 0.85 HPGD (0.57) ALDH1A1SMN1; SMN2KMT2APOLBHTT
SCHEMBL5368197 0.80 TPSAB1 (0.72) MMP13KDM4EPKMF2PLG
SCHEMBL5366075 0.79 MEN1 (0.56) ALDH1A1KMT2APOLBHTTHPGD
SCHEMBL19708998 0.78 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2KMT2APOLBHTT
SCHEMBL14425676 0.77 HTT (0.46) MMP13ALDH1A1SMN1; SMN2KMT2APOLB
SCHEMBL5359305 0.77 KCNH2 (0.73) SMN1; SMN2KMT2A
SCHEMBL6536256 0.76 KDM4E (0.55) KMT2AKDM4EPKMF2PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed