SCHEMBL5370951

SCHEMBL5370951

O=C(NCC1CCN(C(=O)COc2ccc3ccccc3c2)CC1)c1ccc(O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.57
RAB9A P51151 2/20 0.57
NPC1 O15118 1/20 0.57
GPR183 P32249 1/20 0.52
LMNA P02545 1/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
ALOX15 P16050 1/20 0.52
BCHE P06276 1/20 0.52
MAOB P27338 1/20 0.52
ALDH1A1 P00352 3/20 0.50
TP53 P04637 2/20 0.50
USP2 O75604 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367904 0.89 ME2 (0.56) LMNAGAAMAPTALDH1A1USP2
SCHEMBL5362882 0.85 MMP13 (0.56) HPGDALDH1A1TP53USP2SMN1; SMN2
SCHEMBL5366718 0.85 SMN1; SMN2 (0.56) HPGDRAB9AGPR183LMNAMAPT
SCHEMBL5370693 0.85 KMT2A (0.57) RAB9ALMNAGAAMAPTALDH1A1
SCHEMBL5366075 0.81 MEN1 (0.56) HPGDGAAALDH1A1TP53MEN1
SCHEMBL5362915 0.75 HDAC6 (0.60) NPC1POLBHDAC3HDAC4HDAC1
SCHEMBL6536256 0.74 KDM4E (0.55) MEN1KMT2AHDAC3HDAC4HDAC1
SCHEMBL5371009 0.74 PKM (0.51) HPGDRAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL2831262 0.73 NPC1 (0.76) HPGDRAB9ANPC1GPR183LMNA
SCHEMBL5368103 0.72 TPSAB1 (0.71) RAB9ANPC1SMN1; SMN2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed