SCHEMBL5368490

SCHEMBL5368490

O=C(NC(C(=O)C1CC1c1ccccc1F)C1CCNCC1)c1ccnc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 10/20 0.39
KDM1A O60341 1/20 0.38
CDK2 P24941 1/20 0.38
PREP P48147 1/20 0.37
FAP Q12884 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
MAP4K1 Q92918 1/20 0.35
SMYD3 Q9H7B4 2/20 0.35
HDAC4 P56524 1/20 0.34
CSNK1D P48730 1/20 0.34
CSNK1E P49674 1/20 0.34
CHRM1 P11229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5378511 0.90 AKT1 (0.39) AKT1CDK2PREPFAPTAS1R3
SCHEMBL5362652 0.89 AKT1 (0.41) AKT1CDK2PREPFAPTAS1R3
SCHEMBL14425292 0.70 ACHE (0.45) KDM1AHDAC4
SCHEMBL5368483 0.70 ACHE (0.45) KDM1AHDAC4
SCHEMBL5368190 0.68 EPHX2 (0.52) KDM1A
SCHEMBL2859970 0.66 PREP (0.55) PREPFAPTAS1R3TAS1R1TAS1R2
SCHEMBL2860724 0.64 PREP (0.55) PREPFAPTAS1R3TAS1R1TAS1R2
SCHEMBL2860717 0.64 TAS1R3 (0.58) PREPFAPTAS1R3TAS1R1TAS1R2
SCHEMBL2863465 0.63 TAS1R3 (0.57) PREPFAPTAS1R3TAS1R1TAS1R2
SCHEMBL2863458 0.63 TAS1R3 (0.53) PREPFAPTAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed