SCHEMBL5378511

SCHEMBL5378511

O=C(NC(C(=O)C1CC1c1c(F)cccc1F)C1CCNCC1)c1ccnc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 12/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
PREP P48147 1/20 0.38
FAP Q12884 1/20 0.38
CDK2 P24941 1/20 0.36
CHRM1 P11229 1/20 0.36
SMYD3 Q9H7B4 1/20 0.35
MAPT P10636 1/20 0.34
GSK3B P49841 1/20 0.34
ACACB O00763 1/20 0.34
MAP4K1 Q92918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368490 0.90 AKT1 (0.39) AKT1TAS1R3TAS1R1TAS1R2PREP
SCHEMBL5362652 0.88 AKT1 (0.41) AKT1TAS1R3TAS1R1TAS1R2PREP
SCHEMBL5378502 0.69 SIGMAR1 (0.43) GSK3BACACB
SCHEMBL14425293 0.69 SIGMAR1 (0.43) GSK3BACACB
SCHEMBL5366188 0.69 DEGS1 (0.44) AKT1CDK2SMYD3MAPT
SCHEMBL5368190 0.67 EPHX2 (0.52)
SCHEMBL2859970 0.66 PREP (0.55) TAS1R3TAS1R1TAS1R2PREPFAP
SCHEMBL2860717 0.65 TAS1R3 (0.58) TAS1R3TAS1R1TAS1R2PREPFAP
SCHEMBL2860724 0.65 PREP (0.55) TAS1R3TAS1R1TAS1R2PREPFAP
SCHEMBL2863465 0.64 TAS1R3 (0.57) TAS1R3TAS1R1TAS1R2PREPFAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed