SCHEMBL5368519

SCHEMBL5368519

Cc1cc(Cc2ccc(C(F)(F)F)c(Oc3ccc(Cl)cc3)c2)n[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
HTR2A P28223 2/20 0.37
SLC6A4 P31645 2/20 0.37
KCNH2 Q12809 2/20 0.37
RHEB Q15382 1/20 0.35
DAO P14920 3/20 0.35
AR P10275 2/20 0.35
SLC5A2 P31639 1/20 0.35
PLA2G7 Q13093 1/20 0.35
DRD1 P21728 1/20 0.34
PARP1 P09874 1/20 0.34
EGLN1 Q9GZT9 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
ATM Q13315 1/20 0.33
MAPT P10636 2/20 0.33
PPARG P37231 1/20 0.33
PRMT5 O14744 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5385101 0.90 DAO (0.38) CYP3A4CYP2C9CYP2C19DAOAR
SCHEMBL5373755 0.89 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19HTR2ASLC6A4
SCHEMBL5377568 0.84 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19HTR2ASLC6A4
SCHEMBL5375026 0.78 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19HTR2ASLC6A4
SCHEMBL5385763 0.78 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19DAOSLC5A2
SCHEMBL5373734 0.77 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19HTR2ASLC6A4
SCHEMBL5374494 0.74 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19HTR2ASLC6A4
SCHEMBL5365171 0.74 CYP3A4 (0.49) CYP3A4HTR2ASLC6A4KCNH2KDM4E
SCHEMBL5372554 0.74 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19HTR2ASLC6A4
SCHEMBL5374482 0.73 CYP3A4 (0.61) CYP3A4HTR2ASLC6A4KCNH2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed