SCHEMBL5377568

SCHEMBL5377568

O=c1ccc(Cc2ccc(C(F)(F)F)c(Oc3ccc(Cl)cc3)c2)n[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.47
KDR P35968 1/20 0.40
AR P10275 2/20 0.37
HTR2A P28223 3/20 0.36
SLC6A4 P31645 3/20 0.36
KCNH2 Q12809 3/20 0.36
FABP4 P15090 1/20 0.35
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
PLA2G7 Q13093 1/20 0.34
SCN8A Q9UQD0 2/20 0.34
SCN10A Q9Y5Y9 2/20 0.34
CYP2C19 P33261 2/20 0.33
DAO P14920 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
ATM Q13315 1/20 0.33
BRAF P15056 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366909 0.89 CYP3A4 (0.46) CYP3A4KDRTHRATHRBEGLN1
SCHEMBL5374482 0.89 CYP3A4 (0.61) CYP3A4KDRARHTR2ASLC6A4
SCHEMBL5373613 0.85 CYP3A4 (0.51) CYP3A4KDRHTR2ASLC6A4KCNH2
SCHEMBL5368519 0.84 CYP3A4 (0.41) CYP3A4ARHTR2ASLC6A4KCNH2
SCHEMBL5374946 0.84 CYP3A4 (0.42) CYP3A4KDRARSCN8ASCN10A
SCHEMBL5365171 0.83 CYP3A4 (0.49) CYP3A4HTR2ASLC6A4KCNH2FABP4
SCHEMBL5377670 0.82 CYP3A4 (0.48) CYP3A4HTR2ASLC6A4KCNH2CYP2C19
SCHEMBL5421210 0.82 CYP3A4 (0.48) CYP3A4HTR2ASLC6A4KCNH2FABP4
SCHEMBL5373732 0.80 CYP3A4 (0.45) CYP3A4ARKCNH2CYP2C19CYP2C9
SCHEMBL5375034 0.79 CYP3A4 (0.37) CYP3A4KDRARHTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed