SCHEMBL5373755

SCHEMBL5373755

Cc1cc(Cc2ccc(C(F)(F)F)c(Oc3cccc(Cl)c3)c2)n[nH]c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.45
EPAS1 Q99814 1/20 0.41
AR P10275 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
PTGS1 P23219 2/20 0.36
PARP1 P09874 2/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
HTR2A P28223 2/20 0.35
SLC6A4 P31645 2/20 0.35
KCNH2 Q12809 2/20 0.35
PDE5A O76074 1/20 0.35
PDE9A O76083 1/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
TIPARP Q7Z3E1 1/20 0.35
DRD1 P21728 1/20 0.34
NR1H2 P55055 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368519 0.89 CYP3A4 (0.41) CYP3A4ARCYP2C9CYP2C19PARP1
SCHEMBL5385101 0.89 DAO (0.38) CYP3A4ARCYP2C9CYP2C19PARP1
SCHEMBL5374482 0.85 CYP3A4 (0.61) CYP3A4EPAS1ARPTGS1PRMT5
SCHEMBL5375026 0.77 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19PARP1HTR2A
SCHEMBL5385763 0.77 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19PARP1PRMT5
SCHEMBL5374033 0.77 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19PARP1PRMT5
SCHEMBL5386226 0.77 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19PTGS1PRMT5
SCHEMBL5368939 0.76 CYP3A4 (0.64) CYP3A4CYP2C9CYP2C19PTGS1PRMT5
SCHEMBL5368691 0.75 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19PTGS1PARP1
SCHEMBL14570769 0.75 CYP3A4 (0.53) CYP3A4EPAS1CYP2C9CYP2C19PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed