SCHEMBL5368734

SCHEMBL5368734

O=c1ccc(Cc2cccc(OCc3ccc(Cl)cc3)c2)n[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
MEN1 O00255 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NR4A2 P43354 1/20 0.47
MAOA P21397 4/20 0.46
MAOB P27338 4/20 0.46
DPYD Q12882 1/20 0.45
GPR18 Q14330 3/20 0.44
CNR1 P21554 2/20 0.44
CNR2 P34972 1/20 0.44
GPR55 Q9Y2T6 1/20 0.43
HPD P32754 1/20 0.42
SMPD1 P17405 1/20 0.42
TLR4 O00206 1/20 0.42
TLR2 O60603 1/20 0.42
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5375957 0.91 CYP3A4 (0.55) CYP3A4NR4A2MAOAMAOBRXRA
SCHEMBL5367047 0.85 CYP3A4 (0.54) CYP3A4
SCHEMBL5386101 0.84 NR4A2 (0.47) CYP3A4MEN1KMT2ANR4A2MAOA
SCHEMBL5374289 0.81 CYP3A4 (0.64) CYP3A4
SCHEMBL5377482 0.81 CYP3A4 (0.57) CYP3A4
SCHEMBL28778796 0.78 ALPL (0.49) CYP3A4CNR1GPR55
SCHEMBL5377193 0.77 CYP3A4 (0.50) CYP3A4SMN1; SMN2
SCHEMBL5377053 0.77 CYP3A4 (0.51) CYP3A4
SCHEMBL5368812 0.76 CYP3A4 (0.55) CYP3A4
SCHEMBL5373613 0.75 CYP3A4 (0.51) CYP3A4MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed