SCHEMBL5375957

SCHEMBL5375957

O=c1ccc(Cc2cccc(OCc3cccc(Cl)c3)c2)n[nH]1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.55
MAOB P27338 11/20 0.50
MAOA P21397 6/20 0.50
NR4A2 P43354 1/20 0.49
ACHE P22303 1/20 0.46
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368734 0.91 CYP3A4 (0.48) CYP3A4MAOBMAOANR4A2RXRA
SCHEMBL5374289 0.86 CYP3A4 (0.64) CYP3A4
SCHEMBL5386101 0.84 NR4A2 (0.47) CYP3A4MAOBMAOANR4A2
SCHEMBL5367047 0.81 CYP3A4 (0.54) CYP3A4
SCHEMBL5377482 0.81 CYP3A4 (0.57) CYP3A4
SCHEMBL28778796 0.78 ALPL (0.49) CYP3A4
SCHEMBL5377193 0.77 CYP3A4 (0.50) CYP3A4
SCHEMBL5377053 0.77 CYP3A4 (0.51) CYP3A4
SCHEMBL5365181 0.77 CYP3A4 (0.67) CYP3A4
SCHEMBL5368812 0.76 CYP3A4 (0.55) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed