SCHEMBL5375137

SCHEMBL5375137

CSc1ccc(C(=O)c2cc(Cc3ccc(=O)[nH]n3)cc3ccoc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.67
HSD17B10 Q99714 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
PDE4A P27815 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
ATM Q13315 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368514 0.87 CYP3A4 (0.80) CYP3A4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL5365060 0.87 CYP3A4 (0.71) CYP3A4THRATHRBPOLBMAPT
SCHEMBL5373725 0.87 CYP3A4 (0.80) CYP3A4CYP1A2HPGDTHRATHRB
SCHEMBL5369076 0.84 CYP3A4 (0.67) CYP3A4THRATHRBKDM4EPOLB
SCHEMBL5368912 0.83 CYP3A4 (0.83) CYP3A4THRATHRB
SCHEMBL5372475 0.80 CYP3A4 (1.00) CYP3A4HPGDALOX15TSHRPDE4B
SCHEMBL5371101 0.80 CYP3A4 (0.75) CYP3A4HSD17B10ALOX15KDM4EPOLB
SCHEMBL5377729 0.80 CYP3A4 (0.72) CYP3A4THRATHRB
SCHEMBL5365374 0.79 CYP3A4 (0.68) CYP3A4THRATHRBMAPT
SCHEMBL5368780 0.79 CYP3A4 (0.74) CYP3A4CYP1A2THRATHRBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed