SCHEMBL5370356

SCHEMBL5370356

CCC(c1ccc(NC(=O)c2c(Cl)cncc2Cl)cc1)C(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.48
ITGA4 P13612 20/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5146276 1.00 ITGB1 (0.48) ITGB1ITGA4
SCHEMBL5149434 0.88 ITGB1 (0.44) ITGB1ITGA4
SCHEMBL30192895 0.80 PPARG (0.50)
SCHEMBL29231873 0.80 PPARG (0.50)
SCHEMBL2880989 0.79 ITGB1 (0.74) ITGB1ITGA4
SCHEMBL5261609 0.78 ITGB1 (0.54) ITGB1ITGA4
Hydrochloric Acid SCHEMBL5377713 0.77 ITGB1 (0.53) ITGB1ITGA4
Hydrochloric Acid SCHEMBL5149601 0.77 ITGB1 (0.53) ITGB1ITGA4
SCHEMBL1022281 0.77 LMNA (0.46)
SCHEMBL4684731 0.76 CTSK (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291645-B2 Phenylalanine derivatives as alpha 4 integrin inhibitors ELAN PHARMACEUTICALS, INC. (US) 2007-11-06 US disclosed
US-7015216-B2 Heteroaryl-β-alanine derivatives as alpha 4 integrin inhibitors ELAN PHARMACEUTICALS, INC. (US) 2006-03-21 US disclosed
US-6689781-B2 TREATING AN INFLAMMATORY CONDITION IN A MAMMALIAN PATIENT WHICH CONDITION IS MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. 2004-02-10 US disclosed