SCHEMBL5370372

SCHEMBL5370372

Cc1c(Cc2ccc(=O)[nH]n2)ccc(Cl)c1Oc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
THRA P10827 2/20 0.39
THRB P10828 2/20 0.39
RHEB Q15382 2/20 0.35
AKR1B1 P15121 1/20 0.35
NPBWR1 P48145 4/20 0.35
MCHR1 Q99705 1/20 0.35
MAPK8 P45983 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
CNR1 P21554 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5411581 0.88 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5373738 0.87 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5367059 0.86 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5373847 0.74 THRA (0.44) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5364856 0.74 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL4367667 0.74 CYP3A4 (0.53) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5368877 0.73 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19RHEBNPBWR1
SCHEMBL5368441 0.73 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL14570716 0.72 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL17689717 0.71 RHEB (0.44) RHEBNPBWR1MCHR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed