SCHEMBL5372154

SCHEMBL5372154

COc1ccc(C2NC(=S)NC(C)=C2C(C)=O)cc1

nearest known ligand 0.73

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.73
KDM4E B2RXH2 1/20 0.73
TP53 P04637 1/20 0.73
GUSB P08236 1/20 0.70
CA1 P00915 4/20 0.67
CA2 P00918 4/20 0.67
CA12 O43570 1/20 0.64
CA7 P43166 1/20 0.64
CA9 Q16790 1/20 0.64
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
DHFR P00374 2/20 0.59
HTT P42858 1/20 0.57
POLB P06746 1/20 0.54
KMT2A Q03164 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7347481 0.89 GUSB (0.70) ALDH1A1KDM4ETP53GUSBCA1
SCHEMBL7347477 0.89 GUSB (0.70) ALDH1A1KDM4ETP53GUSBCA1
SCHEMBL22639674 0.88 GUSB (0.68) ALDH1A1KDM4ETP53GUSBCA1
SCHEMBL22640045 0.88 GUSB (0.68) ALDH1A1KDM4ETP53GUSBCA1
SCHEMBL28567000 0.84 ALDH1A1 (1.00) ALDH1A1KDM4ETP53CA1CA2
SCHEMBL3168404 0.84 CA1 (0.79) ALDH1A1KDM4EGUSBCA1CA2
SCHEMBL14164074 0.84 DHFR (0.71) ALDH1A1KDM4ETP53GUSBCA1
SCHEMBL14164076 0.82 DHFR (0.72) ALDH1A1KDM4EGUSBCA1CA2
SCHEMBL10113599 0.82 GUSB (1.00) ALDH1A1KDM4ETP53GUSBCA1
SCHEMBL7697757 0.81 CA1 (0.74) ALDH1A1KDM4EGUSBCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160449-B2 Proline chiral columns with broad chiral selectivity VANDERBILT UNIVERSITY (US) 2007-01-09 US disclosed
US-7160449-B2 Proline chiral columns with broad chiral selectivity VANDERBILT UNIVERSITY (US) 2007-01-09 US disclosed
US-7141160-B2 Chiral columns with broad chiral selectivity V{dot over (a)}nderbilt University (US) 2006-11-28 US disclosed
US-20050092686-A1 Proline chiral columns with broad chiral selectivity LI, TINGYU 2005-05-05 US disclosed
EP-0891978-B1 5H-Thiazolo (3,2-a) pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2002-03-20 EP disclosed
EP-0891978-A2 5H-Thiazolo (3,2-a) pyrimidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1999-01-20 EP disclosed