SCHEMBL5373845

SCHEMBL5373845

COc1cc(Cc2ccc(=O)[nH]n2)cc(Oc2cc(C)cc(C)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.40
LMNA P02545 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
AKR1B1 P15121 1/20 0.36
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
THRA P10827 2/20 0.34
THRB P10828 2/20 0.34
ALDH1A1 P00352 2/20 0.33
ALPL P05186 1/20 0.33
HTT P42858 1/20 0.33
NPBWR1 P48145 1/20 0.33
IDH1 O75874 1/20 0.33
CALM1 P0DP23 1/20 0.33
CYP19A1 P11511 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5376945 0.88 CYP3A4 (0.44) CYP3A4LMNASMN1; SMN2NPC1PDE4B
SCHEMBL5374014 0.86 CYP3A4 (0.48) CYP3A4LMNASMN1; SMN2NPC1RAB9A
SCHEMBL5377730 0.85 CYP3A4 (0.45) CYP3A4LMNASMN1; SMN2NPC1RAB9A
SCHEMBL5375921 0.84 CYP3A4 (0.48) CYP3A4LMNASMN1; SMN2NPC1RAB9A
SCHEMBL5375382 0.83 CYP3A4 (0.45) CYP3A4SMN1; SMN2NPC1RAB9AAKR1B1
SCHEMBL5372571 0.80 CYP3A4 (0.60) CYP3A4AKR1B1
SCHEMBL5369070 0.79 CYP3A4 (0.47) CYP3A4NPC1ALDH1A1ALPLHTT
SCHEMBL28778796 0.78 ALPL (0.49) CYP3A4LMNAALPLIDH1
SCHEMBL5372604 0.75 CYP3A4 (0.71) CYP3A4LMNANPC1RAB9ATHRA
SCHEMBL5373837 0.75 CYP3A4 (0.47) CYP3A4LMNANPC1THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed