Sch-58261

Sch-58261

SCHEMBL537287

Nc1nc2c(cnn2CCc2ccccc2)c2nc(-c3ccco3)nn12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 15/20 1.00
ADORA1 P30542 9/20 1.00
KDM4E B2RXH2 1/20 1.00
NPC1 O15118 1/20 1.00
ALDH1A1 P00352 1/20 1.00
TP53 P04637 1/20 1.00
CYP3A4 P08684 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
HPGD P15428 1/20 1.00
ALOX15 P16050 1/20 1.00
MAPK1 P28482 1/20 1.00
ADORA2B P29275 1/20 1.00
RAB9A P51151 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
HSD17B10 Q99714 1/20 1.00
HDAC1 Q13547 1/20 0.75
HDAC6 Q9UBN7 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sch-63390 SCHEMBL5823548 0.94 ADORA2A (1.00) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL7345461 0.91 ADORA2A (1.00) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL22796280 0.91 ADORA2A (0.85) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL20694157 0.91 ADORA2A (0.85) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL7339226 0.91 ADORA2A (1.00) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL23691785 0.91 ADORA2A (0.85) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL21588751 0.90 ADORA2A (0.90) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL14922365 0.88 ADORA2A (0.86) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL7336459 0.88 ADORA2A (0.81) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL21588752 0.88 ADORA2A (0.78) ADORA2AADORA1KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 972 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250213684-A1 COMBINATION THERAPIES COMPRISING ANTIBODY MOLECULES TO TIM-3 NOVARTIS AG (CH) 2025-07-03 US claimed
US-20250161313-A1 A METHOD FOR THE TREATMENT OF NEUROPATHY Institut National de la Santé et de la Recherche Médicale (FR) 2025-05-22 US claimed
US-20250161312-A1 A METHOD FOR THE TREATMENT OF CHEMOTHERAPEUTIC DRUG-INDUCED NEPHROTOXICITY Institut National de la Santé et de la Recherche Médicale (FR) 2025-05-22 US claimed
US-12303618-B2 Oxygen-generating cryogels NORTHEASTERN UNIVERSITY (US) 2025-05-20 US claimed
CN-119969964-A Research method for influence on TBI post-impulse behavior 重庆医科大学 2025-05-13 CN claimed
EP-4489759-A1 A METHOD FOR THE TREATMENT OF NEUROPATHY Institut National de la Santé et de la Recherche Médicale (INSERM) (FR) 2025-01-15 EP claimed
EP-4489760-A1 A METHOD FOR THE TREATMENT OF CHEMOTHERAPEUTIC DRUG-INDUCED NEPHROTOXICITY Institut National de la Santé et de la Recherche Médicale (INSERM) (FR) 2025-01-15 EP claimed
WO-2024216134-A1 COMBINATORIAL STRATEGIES TO ENHANCE VACCINIA VIRUS IN VITRO AND IN VIVO ONCOLYSIS UNIVERSITY OF MIAMI (US) 2024-10-17 WO claimed
US-20240219394-A1 METHOD FOR MEASURING RESPONSE OF OLFACTORY RECEPTOR TO SUBSTANCE AJINOMOTO CO., INC. (JP) 2024-07-04 US claimed
EP-4382612-A1 METHOD FOR MEASURING RESPONSE OF OLFACTORY RECEPTOR TO SUBSTANCE AJINOMOTO CO., INC. (JP) 2024-06-12 EP claimed
US-20160151374-A1 METHOD OF USING VASOCONSTRICTIVE AGENTS DURING ENERGY-BASED TISSUE THERAPY SHERWOOD SERVICES AG (CH) 2016-06-02 US claimed
US-9271985-B2 Method of using vasoconstrictive agents during energy-based tissue therapy COVIDIEN AG (CH) 2016-03-01 US claimed
US-20150164903-A1 METHOD OF USING VASOCONSTRICTIVE AGENTS DURING ENERGY-BASED TISSUE THERAPY SHERWOOD SERVICES AG (CH) 2015-06-18 US claimed
US-20140271606-A1 METHODS OF USING ADENOSINE RECEPTOR ANTAGONISTS FOR TREATING BLEEDING DISORDERS BAYER HEALTHCARE LLC 2014-09-18 US claimed
US-7767686-B2 Method of using adenosine receptor blockers during tissue ablation COVIDIEN AG (CH) 2010-08-03 US claimed
US-20080275068-A1 administering a vasoconstrictive agent such as an adenosine receptor antagonist ( 1,3-dipropyl-8-cyclopentylxanthine, 8-(3-Chlorostyryl)caffeine, 6-carboxy-methyl-5,9-dihydro-9-methyl-2-phenyl-[1,2,4]-triazolo[5,1-a][2,7]naphthyridine) to the mammal to increases the size of the coagulation zone COVIDIEN AG (CH) 2008-11-06 US claimed
US-20070208042-A1 Method of using vasoconstrictive agents during energy-based tissue therapy SHERWOOD SERVICES AG 2007-09-06 US claimed
US-20070207979-A1 Method of using adenosine receptor blockers during tissue ablation SHERWOOD SERVICES AG 2007-09-06 US claimed
EP-1300147-A1 Purine compounds and adenosine A2 receptor antagonist as preventive or therapeutic agent for diabetes mellitus Eisai Co. Ltd (JP) 2003-04-09 EP claimed
EP-1054012-A1 PURINE DERIVATIVES AND ADENOSINE A2 RECEPTOR ANTAGONISTS SERVING AS PREVENTIVES/REMEDIES FOR DIABETES Eisai Co., Ltd. (JP) 2000-11-22 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250161313-A1 A METHOD FOR THE TREATMENT OF NEUROPATHY ADORA2A, P2RX2, ADORA2B ADORA2A 1/4885ADORA1 12/4885KDM4E 1434/4885
US-20070207979-A1 Method of using adenosine receptor blockers during tissue ablation ADORA2A, ADORA2B, ADORA3 ADORA2A 1/4885ADORA1 4/4885KDM4E 4216/4885
US-20250213684-A1 COMBINATION THERAPIES COMPRISING ANTIBODY MOLECULES TO TIM-3 HAVCR2, LGALS3BP, CD274 ADORA2A 1416/4885ADORA1 2549/4885KDM4E 3970/4885
US-20070208042-A1 Method of using vasoconstrictive agents during energy-based tissue therapy PLAT, TEK, PLG ADORA2A 271/4885ADORA1 503/4885KDM4E 3340/4885
US-20250161312-A1 A METHOD FOR THE TREATMENT OF CHEMOTHERAPEUTIC DRUG-INDUCED NEPHROTOXICITY ADORA2A, ADORA3, ADORA2B ADORA2A 1/4885ADORA1 5/4885KDM4E 1738/4885
US-20150164903-A1 METHOD OF USING VASOCONSTRICTIVE AGENTS DURING ENERGY-BASED TISSUE THERAPY PLAT, TEK, PLG ADORA2A 271/4885ADORA1 503/4885KDM4E 3340/4885
US-20160151374-A1 METHOD OF USING VASOCONSTRICTIVE AGENTS DURING ENERGY-BASED TISSUE THERAPY PLAT, TEK, PLG ADORA2A 271/4885ADORA1 503/4885KDM4E 3340/4885
US-20080275068-A1 administering a vasoconstrictive agent such as an adenosine receptor antagonist ( 1,3-dipropyl-8-cyclopentylxanthine, 8-(3-Chlorostyryl)caffeine, 6-carboxy-methyl-5,9-dihydro-9-methyl-2-phenyl-[1,2,4]-triazolo[5,1-a][2,7]naphthyridine) to the mammal to increases the size of the coagulation zone ADORA2A, ADORA1, ADORA3 ADORA2A 1/4885ADORA1 2/4885KDM4E 1872/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.