SCHEMBL5373967

SCHEMBL5373967

O=c1ccc(Cc2cc(Cc3ccc(Cl)cc3)c3ccccc3c2)n[nH]1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.54
PTGS2 P35354 1/20 0.46
LMNA P02545 2/20 0.44
DAO P14920 6/20 0.40
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PRNP P04156 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373636 0.81 CYP3A4 (0.56) CYP3A4PTGS2LMNADAOMAPT
SCHEMBL5374280 0.78 CYP3A4 (0.50) CYP3A4LMNA
SCHEMBL5382621 0.77 CYP3A4 (0.54) CYP3A4DAO
SCHEMBL5375840 0.73 CYP3A4 (0.55) CYP3A4DAO
SCHEMBL5373848 0.72 CYP3A4 (0.54) CYP3A4
SCHEMBL5351260 0.72 AKR1B1 (0.51) CYP3A4LMNADAO
SCHEMBL5381870 0.72 CYP3A4 (0.48) CYP3A4DAO
SCHEMBL5367220 0.71 CYP3A4 (0.84) CYP3A4
SCHEMBL5368836 0.71 CYP3A4 (0.64) CYP3A4DAOMAPT
SCHEMBL5373933 0.68 CYP3A4 (0.45) CYP3A4LMNADAOMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed