SCHEMBL5374014

SCHEMBL5374014

COc1cc(Cc2ccc(=O)[nH]n2)cc(Oc2cc(Cl)cc(Cl)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.48
LMNA P02545 2/20 0.38
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
AKR1B1 P15121 1/20 0.35
TOP2A P11388 2/20 0.35
KDM4E B2RXH2 1/20 0.34
GRK6 P43250 1/20 0.34
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
KMT2A Q03164 1/20 0.33
FAAH O00519 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377730 0.92 CYP3A4 (0.45) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL5368755 0.88 CYP3A4 (0.47) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL5375921 0.88 CYP3A4 (0.48) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL5373999 0.88 CYP3A4 (0.48) CYP3A4LMNANPC1RAB9AAKR1B1
SCHEMBL5376945 0.86 CYP3A4 (0.44) CYP3A4LMNANPC1SMN1; SMN2KDM4E
SCHEMBL5373845 0.86 CYP3A4 (0.40) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL5377482 0.84 CYP3A4 (0.57) CYP3A4THRATHRBFAAH
SCHEMBL14559652 0.82 CYP3A4 (0.51) CYP3A4LMNASMN1; SMN2PDE4APDE4B
SCHEMBL5370922 0.80 CYP3A4 (0.45) CYP3A4NPC1RAB9ASMN1; SMN2AKR1B1
SCHEMBL5375382 0.80 CYP3A4 (0.45) CYP3A4NPC1RAB9ASMN1; SMN2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed