SCHEMBL14559652

SCHEMBL14559652

COc1ccc(Cc2ccc(=O)[nH]n2)cc1Oc1cc(Cl)cc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.43
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
CYP2C9 P11712 2/20 0.41
TSHR P16473 2/20 0.41
CYP2C19 P33261 2/20 0.41
CA2 P00918 1/20 0.39
POLB P06746 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 2/20 0.37
MPI P34949 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
PDE3B Q13370 2/20 0.37
PDE3A Q14432 2/20 0.37
CCNE2 O96020 1/20 0.36
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377670 0.91 CYP3A4 (0.48) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5368714 0.87 CYP3A4 (0.53) CYP3A4SMN1; SMN2ALDH1A1KMT2ADAO
SCHEMBL5365424 0.86 CYP3A4 (0.48) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5370279 0.86 CYP3A4 (0.53) CYP3A4SMN1; SMN2ALDH1A1KMT2ADAO
SCHEMBL5374014 0.82 CYP3A4 (0.48) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5382226 0.81 CACNA1G (0.44) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5370543 0.79 CYP3A4 (0.46) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5377482 0.79 CYP3A4 (0.57) CYP3A4
SCHEMBL5365171 0.78 CYP3A4 (0.49) CYP3A4SMN1; SMN2LMNA
SCHEMBL5386025 0.78 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19CCNE2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed