SCHEMBL5377730

SCHEMBL5377730

COc1cc(Cc2ccc(=O)[nH]n2)cc(Oc2ccc(Cl)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
LMNA P02545 2/20 0.40
TOP2A P11388 1/20 0.39
NPBWR1 P48145 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
AKR1B1 P15121 1/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
MAPT P10636 2/20 0.36
CNR1 P21554 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
LTA4H P09960 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
OPRK1 P41145 1/20 0.35
FAAH O00519 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374014 0.92 CYP3A4 (0.48) CYP3A4LMNATOP2ANPC1RAB9A
SCHEMBL5370922 0.88 CYP3A4 (0.45) CYP3A4NPC1RAB9ASMN1; SMN2AKR1B1
SCHEMBL5375382 0.88 CYP3A4 (0.45) CYP3A4NPBWR1NPC1RAB9ASMN1; SMN2
SCHEMBL5376945 0.88 CYP3A4 (0.44) CYP3A4LMNANPC1SMN1; SMN2LTA4H
SCHEMBL5373845 0.85 CYP3A4 (0.40) CYP3A4LMNANPBWR1NPC1RAB9A
SCHEMBL5367047 0.83 CYP3A4 (0.54) CYP3A4LMNAFAAHALDH1A1
SCHEMBL5377670 0.81 CYP3A4 (0.48) CYP3A4LMNANPBWR1SMN1; SMN2MAPT
SCHEMBL5368755 0.80 CYP3A4 (0.47) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL5373999 0.80 CYP3A4 (0.48) CYP3A4LMNANPC1RAB9AAKR1B1
SCHEMBL5375921 0.80 CYP3A4 (0.48) CYP3A4LMNANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed