SCHEMBL5374431

SCHEMBL5374431

CC[C@@H](N)CC#N.O=C(OC(C(=O)O)C(OC(=O)c1ccccc1)C(=O)O)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.59
TP53 P04637 1/20 0.59
CYP2D6 P10635 3/20 0.48
RECQL P46063 1/20 0.46
LMNA P02545 3/20 0.39
CYP1A2 P05177 2/20 0.38
POLB P06746 1/20 0.38
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
NPC1 O15118 3/20 0.37
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
ALDH1A1 P00352 2/20 0.36
SLC1A5 Q15758 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565308 1.00 TSHR (0.59) TSHRTP53CYP2D6RECQLLMNA
SCHEMBL6229562 1.00 TSHR (0.59) TSHRTP53CYP2D6RECQLLMNA
SCHEMBL5388738 1.00 TSHR (0.59) TSHRTP53CYP2D6RECQLLMNA
SCHEMBL5378640 0.90 TP53 (0.45) TSHRTP53CYP2D6RECQLLMNA
Alcohol SCHEMBL18886336 0.81 TSHR (0.79) TSHRTP53CYP2D6RECQLLMNA
SCHEMBL2596645 0.80 TSHR (0.58) TSHRTP53CYP2D6RECQLLMNA
SCHEMBL5867194 0.80 TSHR (0.58) TSHRTP53CYP2D6RECQLLMNA
Water SCHEMBL365251 0.79 TSHR (0.96) TSHRTP53CYP2D6RECQLLMNA
Water SCHEMBL312080 0.79 TSHR (0.96) TSHRTP53CYP2D6RECQLLMNA
Water SCHEMBL2859440 0.79 TSHR (0.96) TSHRTP53CYP2D6RECQLLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7301044-B2 Preparation of chiral amino-nitriles PFIZER INC. (US) 2007-11-27 US claimed
EP-1517877-A1 PREPARATION OF CHIRAL AMINO-NITRILES PCBU Services, Inc. (US) 2005-03-30 EP claimed
US-20050038281-A1 Preparation of chiral amino-nitriles PFIZER INC. 2005-02-17 US claimed
WO-2004002924-A1 PREPARATION OF CHIRAL AMINO-NITRILES PCBU SERVICES, INC. (US) 2004-01-08 WO claimed
US-20040002615-A1 PREPARATION OF CHIRAL AMINO-NITRILES PFIZER INC. 2004-01-01 US claimed
US-7301044-B2 Preparation of chiral amino-nitriles PFIZER INC. (US) 2007-11-27 US disclosed
EP-1517877-A1 PREPARATION OF CHIRAL AMINO-NITRILES PCBU Services, Inc. (US) 2005-03-30 EP disclosed
US-20050038281-A1 Preparation of chiral amino-nitriles PFIZER INC. 2005-02-17 US disclosed
WO-2004002924-A1 PREPARATION OF CHIRAL AMINO-NITRILES PCBU SERVICES, INC. (US) 2004-01-08 WO disclosed
US-20040002615-A1 PREPARATION OF CHIRAL AMINO-NITRILES PFIZER INC. 2004-01-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038281-A1 Preparation of chiral amino-nitriles NOS3, NOS1, NOS2 TSHR 4098/4885TP53 3927/4885CYP2D6 684/4885
US-20040002615-A1 PREPARATION OF CHIRAL AMINO-NITRILES NOS3, NOS1, NOS2 TSHR 4098/4885TP53 3927/4885CYP2D6 684/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.