SCHEMBL5374877

SCHEMBL5374877

CCOC(=O)/C=C/c1cn(Cc2ccc(OCc3ccccc3)cc2)cc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
LMNA P02545 2/20 0.44
PPARG P37231 1/20 0.44
BACE1 P56817 2/20 0.43
S1PR5 Q9H228 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
PTPN1 P18031 1/20 0.43
ALDH1A1 P00352 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HDAC8 Q9BY41 1/20 0.41
PTGS1 P23219 2/20 0.41
PTGS2 P35354 2/20 0.41
ALOX5 P09917 2/20 0.41
GSK3B P49841 1/20 0.41
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5385296 0.92 PTGER3 (0.48) NR1H4PPARGBACE1HDAC8ALOX5
SCHEMBL5377058 0.91 BACE1 (0.43) NR1H4L3MBTL1LMNAPPARGBACE1
SCHEMBL6592132 0.87 PTGER3 (0.51) BACE1S1PR5ALDH1A1PTGS1PTGS2
SCHEMBL6592125 0.87 PTGER3 (0.51) BACE1S1PR5ALDH1A1PTGS1PTGS2
SCHEMBL5387806 0.86 FFAR1 (0.55) PPARG
SCHEMBL5397126 0.82 GAA (0.61) NR1H4L3MBTL1LMNAPTGDR2ALDH1A1
SCHEMBL5385879 0.81 KMT2A (0.47) L3MBTL1LMNAPPARGALDH1A1SMN1; SMN2
SCHEMBL6595111 0.80 PTGER3 (0.61) BACE1ALDH1A1PTGS1PTGS2ALOX5
SCHEMBL6595113 0.80 PTGER3 (0.61) BACE1ALDH1A1PTGS1PTGS2ALOX5
SCHEMBL5374881 0.80 LTB4R (0.47) NR1H4L3MBTL1PPARGS1PR5PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179823-B1 5-membered n-heterocyclic compounds with hypoglycemic and hypolipidemic activity TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-20 US disclosed