SCHEMBL5375017

SCHEMBL5375017

O=c1ccc(Cc2ccc(F)c(Oc3ccccc3)c2)n[nH]1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.51
DAO P14920 2/20 0.39
PARP1 P09874 3/20 0.39
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
AKR1B1 P15121 2/20 0.34
TTR P02766 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377723 0.89 CYP3A4 (0.66) CYP3A4DAOPARP1AKR1B1CYP2C9
SCHEMBL5377473 0.88 CYP3A4 (0.52) CYP3A4PARP1THRATHRBAKR1B1
SCHEMBL5370279 0.87 CYP3A4 (0.53) CYP3A4DAOPARP1THRATHRB
SCHEMBL5365456 0.86 CYP3A4 (0.50) CYP3A4PARP1AKR1B1
SCHEMBL5368917 0.85 CYP3A4 (0.48) CYP3A4DAOTHRATHRBAKR1B1
SCHEMBL4367667 0.85 CYP3A4 (0.53) CYP3A4DAOTHRATHRBAKR1B1
SCHEMBL5370985 0.85 CYP3A4 (0.48) CYP3A4DAOPARP1THRATHRB
SCHEMBL5374410 0.85 CYP3A4 (0.49) CYP3A4PARP1
SCHEMBL5366909 0.85 CYP3A4 (0.46) CYP3A4DAOTHRATHRBAKR1B1
SCHEMBL5377719 0.85 CYP3A4 (0.46) CYP3A4PARP1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed