SCHEMBL5366909

SCHEMBL5366909

O=c1ccc(Cc2ccc(C(F)(F)F)c(Oc3ccccc3)c2)n[nH]1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
NTRK1 P04629 1/20 0.38
AKR1B1 P15121 3/20 0.37
KDR P35968 1/20 0.35
DAO P14920 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
EGLN1 Q9GZT9 1/20 0.33
LPAR1 Q92633 1/20 0.33
LPAR5 Q9H1C0 1/20 0.33
ENPP1 P22413 1/20 0.33
MGLL Q99685 1/20 0.33
NR3C1 P04150 1/20 0.32
FDFT1 P37268 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377568 0.89 CYP3A4 (0.47) CYP3A4KDRDAOSCN8ASCN10A
SCHEMBL5374482 0.88 CYP3A4 (0.61) CYP3A4AKR1B1KDR
SCHEMBL5374946 0.86 CYP3A4 (0.42) CYP3A4NTRK1AKR1B1KDRDAO
SCHEMBL5373732 0.86 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19
SCHEMBL5375017 0.85 CYP3A4 (0.51) CYP3A4AKR1B1DAOTHRATHRB
SCHEMBL5385101 0.84 DAO (0.38) CYP3A4DAOENPP1MGLLCYP2C9
SCHEMBL5368699 0.83 AR (0.39) CYP3A4AKR1B1
SCHEMBL5370985 0.82 CYP3A4 (0.48) CYP3A4DAOTHRATHRBCYP2C9
SCHEMBL5368917 0.82 CYP3A4 (0.48) CYP3A4NTRK1AKR1B1DAOTHRA
SCHEMBL4367667 0.82 CYP3A4 (0.53) CYP3A4AKR1B1DAOTHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed