SCHEMBL5375203

SCHEMBL5375203

O=c1cc(-c2ccncc2)[nH]c(Cc2ccc(Cl)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.47
GCGR P47871 8/20 0.46
MAPK14 Q16539 5/20 0.46
ROCK2 O75116 1/20 0.40
GRK2 P25098 1/20 0.40
CDC7 O00311 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5386993 0.88 GSK3B (0.48) GSK3BGCGRMAPK14CDC7
SCHEMBL5376093 0.86 GSK3B (0.63) GSK3BMAPK14CDC7
SCHEMBL5390451 0.84 GSK3B (0.45) GSK3BGCGRMAPK14CDC7
SCHEMBL5382412 0.83 CYP3A4 (0.41) GSK3BGCGRMAPK14ROCK2
SCHEMBL5381458 0.83 CYP17A1 (0.47) GSK3BGCGRMAPK14CDC7
SCHEMBL5382469 0.82 GSK3B (0.49) GSK3BGCGRCDC7
SCHEMBL5386907 0.82 GSK3B (0.48) GSK3BCDC7
SCHEMBL5376071 0.80 GSK3B (0.49) GSK3BCDC7
SCHEMBL5380257 0.79 MAPT (0.49) GSK3BCDC7
SCHEMBL5390690 0.79 GSK3B (0.48) GSK3BMAPK14ROCK2CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP claimed
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP claimed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO claimed
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed