Cefoperazone

Cefoperazone

SCHEMBL537680

CCN1CCN(C(=O)N[C@@H](C(=O)N[C@@H]2C(=O)N3C(C(=O)[O-])=C(CSc4nnnn4C)CS[C@H]23)c2ccc(O)cc2)C(=O)C1=O.[Na+]

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Cefoperazone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 9/20 1.00
MAPT P10636 10/20 0.88
SLC22A6 Q4U2R8 2/20 0.88
SLC22A8 Q8TCC7 2/20 0.88
SLC22A11 Q9NSA0 2/20 0.88
PDE3A Q14432 1/20 0.88
HSD17B10 Q99714 5/20 0.87
THRB P10828 1/20 0.87
TSHR P16473 1/20 0.87
POLB P06746 8/20 0.63
ALDH1A1 P00352 5/20 0.63
CYP3A4 P08684 2/20 0.63
KDM4E B2RXH2 1/20 0.63
HPGD P15428 1/20 0.63
APEX1 P27695 1/20 0.63
PTPN7 P35236 1/20 0.63
NR1I2 O75469 1/20 0.54
PGR P06401 1/20 0.54
PPARG P37231 1/20 0.54
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11089531 0.94 TDP1 (0.90) TDP1MAPTSLC22A6SLC22A8SLC22A11
SCHEMBL11083504 0.94 TDP1 (0.90) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL6655255 0.94 MAPT (0.99) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL11522109 0.94 MAPT (1.00) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL18061225 0.94 MAPT (1.00) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL16072819 0.94 MAPT (1.00) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL15387468 0.94 MAPT (1.00) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL2222952 0.94 MAPT (1.00) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL16091123 0.94 MAPT (1.00) TDP1MAPTSLC22A6SLC22A8SLC22A11
Cefoperazone SCHEMBL9326569 0.94 MAPT (1.00) TDP1MAPTSLC22A6SLC22A8SLC22A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 255 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116687867-A Cefoperazone sodium for injection and preparation method thereof 南京恩泰医药科技有限公司 2023-09-05 CN claimed
US-9227999-B2 Antimicrobial cationic peptides and formulations thereof CARRUS CAPITAL CORPORATION (CA) 2016-01-05 US claimed
US-20260027191-A1 COMPOSITIONS AND METHODS FOR TREATING BACTERIAL DISEASE UNIV ARIZONA (US) 2026-01-29 US disclosed
EP-3866826-B1 ANTIMICROBIAL PEPTIDES AND METHODS OF USING THE SAME RIPTIDE BIOSCIENCE INC (US) 2025-12-10 EP disclosed
EP-4628100-A2 ANTI-VIRAL COMPOUNDS AND METHODS FOR ADMINISTRATION THEREOF Gregg, John Malcolm Hall (US) 2025-10-08 EP disclosed
US-12285413-B2 Anti-viral agents and methods for administration thereof GREGG JOHN M H (US) 2025-04-29 US disclosed
CN-119818504-A Antibacterial composition of cefoperazone and avibactam and application thereof 重庆圣华曦药业股份有限公司 2025-04-15 CN disclosed
CN-113861268-B Cell penetrating peptides and methods of making and using the same 恩特拉达治疗学股份有限公司 2025-04-01 CN disclosed
US-20250099566-A1 COMPOSITIONS AND METHODS FOR TREATING BACTERIAL DISEASE NATIONAL INSTITUTES OF HEALTH 2025-03-27 US disclosed
WO-2025059113-A1 TREATMENTS FOR ENHANCING IMMUNE RESPONSE TO CLOSTRIDIOIDES DIFFICILE INFECTIONS THE BOARD OF REGENTS OF THE UNIVERSITY OF OKLAHOMA (US) 2025-03-20 WO disclosed
CN-119391643-B Culture medium and method for culturing digestive tract tumor by using three-dimensional tumor tablet technology 珠海澳大科技研究院 2025-03-14 CN disclosed
EP-0925308-B1 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING ANALOGUES OF INDOLICIDIN MICROLOGIX BIOTECH INC (CA) 2002-06-05 EP disclosed
US-20020035061-A1 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING CATIONIC PEPTIDES ALONE OR IN COMBINATION WITH ANTIBIOTICS BIOWEST THERAPEUTICS INC. (CA) 2002-03-21 US disclosed
EP-1174439-A2 Compositions and methods for treating infections using analogues of indolicidin Micrologix Biotech, Inc. (CA) 2002-01-23 EP disclosed
US-6180604-B1 Compositions and methods for treating infections using analogues of indolicidin MICROLOGIX BIOTECH INC. (CA) 2001-01-30 US disclosed
EP-0966481-A2 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING CATIONIC PEPTIDES ALONE OR IN COMBINATION WITH ANTIBIOTICS Micrologix Biotech, Inc. (CA) 1999-12-29 EP disclosed
EP-0925308-A2 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING ANALOGUES OF INDOLICIDIN Micrologix Biotech, Inc. (CA) 1999-06-30 EP disclosed
WO-1998040401-A2 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING CATIONIC PEPTIDES ALONE OR IN COMBINATION WITH ANTIBIOTICS MICROLOGIX BIOTECH INC. (CA) 1998-09-17 WO disclosed
WO-1998007745-A9 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING ANALOGUES OF INDOLICIDIN 1998-04-23 WO disclosed
WO-1998007745-A2 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING ANALOGUES OF INDOLICIDIN MICROLOGIX BIOTECH, INC. (CA) 1998-02-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260027191-A1 COMPOSITIONS AND METHODS FOR TREATING BACTERIAL DISEASE DNMT3L, DNMT3A, DNMT1 TDP1 236/4885MAPT 2164/4885SLC22A6 305/4885
US-12285413-B2 Anti-viral agents and methods for administration thereof ACE2, ACE, MAVS TDP1 2443/4885MAPT 2631/4885SLC22A6 942/4885
US-20020035061-A1 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS USING CATIONIC PEPTIDES ALONE OR IN COMBINATION WITH ANTIBIOTICS VIP, PEPD, PTMS TDP1 3303/4885MAPT 2784/4885SLC22A6 3082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.