SCHEMBL5377358

SCHEMBL5377358

CCOC(=O)CCc1cn(Cc2ccc(OCc3csc(-c4cccnc4)n3)cc2)cc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.46
MAPT P10636 2/20 0.46
POLB P06746 2/20 0.46
ALDH1A1 P00352 5/20 0.43
DNM1L O00429 2/20 0.41
PDE10A Q9Y233 1/20 0.41
MMP13 P45452 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
RAB9A P51151 3/20 0.39
KDM4E B2RXH2 2/20 0.38
GAA P10253 1/20 0.38
CPT1A P50416 1/20 0.38
CPT1B Q92523 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
NPC1 O15118 2/20 0.38
NFKB1 P19838 2/20 0.38
NFKB2 Q00653 2/20 0.38
RELA Q04206 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5385880 0.94 ALDH1A1 (0.46) TP53MAPTPOLBALDH1A1MMP13
SCHEMBL5377258 0.94 ALDH1A1 (0.48) TP53MAPTPOLBALDH1A1SMN1; SMN2
SCHEMBL5382597 0.91 ALDH1A1 (0.41) TP53MAPTPOLBALDH1A1MMP13
SCHEMBL5377468 0.91 TP53 (0.44) TP53MAPTPOLBALDH1A1DNM1L
SCHEMBL5374473 0.89 ALDH1A1 (0.42) TP53MAPTALDH1A1SMN1; SMN2RAB9A
SCHEMBL5372016 0.88 L3MBTL1 (0.42) ALDH1A1SMN1; SMN2RAB9AGAAL3MBTL1
SCHEMBL5381657 0.87 ALDH1A1 (0.42) TP53MAPTPOLBALDH1A1SMN1; SMN2
SCHEMBL5385582 0.87 ALDH1A1 (0.44) TP53MAPTALDH1A1SMN1; SMN2RAB9A
SCHEMBL5377265 0.86 ALDH1A1 (0.41) TP53MAPTPOLBALDH1A1SMN1; SMN2
SCHEMBL5397102 0.86 ALDH1A1 (0.46) TP53MAPTPOLBALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179823-B1 5-membered n-heterocyclic compounds with hypoglycemic and hypolipidemic activity TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-20 US disclosed
EP-1457490-A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity Takeda Chemical Industries, Ltd. (JP) 2004-09-15 EP disclosed
EP-1228067-B1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-07-14 EP disclosed