SCHEMBL5377627

SCHEMBL5377627

O=c1ccc(Cc2ccc(Br)c(Oc3cccc(Cl)c3)c2)n[nH]1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.64
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
SLC6A4 P31645 4/20 0.37
AKR1B1 P15121 1/20 0.36
HTR2A P28223 1/20 0.36
KCNH2 Q12809 1/20 0.36
AHR P35869 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
RHEB Q15382 3/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A3 Q01959 2/20 0.34
HTR1A P08908 1/20 0.34
MAPK8 P45983 1/20 0.34
FAAH O00519 1/20 0.34
P2RX4 Q99571 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365181 0.89 CYP3A4 (0.67) CYP3A4SLC6A4AKR1B1HTR2AKCNH2
SCHEMBL5377723 0.88 CYP3A4 (0.66) CYP3A4SLC6A4AKR1B1HTR2AKCNH2
SCHEMBL5368917 0.88 CYP3A4 (0.48) CYP3A4THRATHRBAKR1B1
SCHEMBL5368939 0.87 CYP3A4 (0.64) CYP3A4SLC6A4AKR1B1HTR2AKCNH2
SCHEMBL5370245 0.86 CYP3A4 (0.63) CYP3A4THRATHRBSLC6A4AKR1B1
SCHEMBL5372601 0.85 CYP3A4 (0.62) CYP3A4THRATHRBSLC6A4AKR1B1
SCHEMBL5374289 0.85 CYP3A4 (0.64) CYP3A4AKR1B1AHRPRMT5WDR77
SCHEMBL5374482 0.84 CYP3A4 (0.61) CYP3A4SLC6A4AKR1B1HTR2AKCNH2
SCHEMBL5370328 0.84 CYP3A4 (0.47) CYP3A4THRATHRBFNTAFNTB
SCHEMBL5374390 0.83 CYP3A4 (0.46) CYP3A4THRATHRBAKR1B1RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed