SCHEMBL5377670

SCHEMBL5377670

COc1ccc(Cc2ccc(=O)[nH]n2)cc1Oc1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.43
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 3/20 0.39
CA2 P00918 1/20 0.39
RECQL P46063 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 2/20 0.38
GAA P10253 2/20 0.37
LMNA P02545 2/20 0.37
USP2 O75604 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
POLB P06746 1/20 0.37
MPI P34949 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14559652 0.91 CYP3A4 (0.51) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5365424 0.88 CYP3A4 (0.48) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5365171 0.87 CYP3A4 (0.49) CYP3A4SMN1; SMN2LMNAHTR2ASLC6A4
SCHEMBL5373613 0.87 CYP3A4 (0.51) CYP3A4LMNAHTR2ASLC6A4KCNH2
SCHEMBL5421210 0.86 CYP3A4 (0.48) CYP3A4LMNAHTR2ASLC6A4KCNH2
SCHEMBL5382226 0.86 CACNA1G (0.44) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5377568 0.82 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19HTR2ASLC6A4
SCHEMBL5377730 0.81 CYP3A4 (0.45) CYP3A4SMN1; SMN2ALDH1A1MAPTLMNA
SCHEMBL5370543 0.79 CYP3A4 (0.46) CYP3A4SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL5367047 0.79 CYP3A4 (0.54) CYP3A4ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed