SCHEMBL5378297

SCHEMBL5378297

Cc1nc(Cl)c(N2CCC(O)C2)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.34
NPY5R Q15761 1/20 0.34
SLC34A1 Q06495 1/20 0.33
RAD52 P43351 1/20 0.33
METAP2 P50579 4/20 0.33
SLC6A3 Q01959 2/20 0.33
GABRA1 P14867 1/20 0.33
SMO Q99835 2/20 0.33
CHRM3 P20309 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
CNR2 P34972 4/20 0.32
PRKDC P78527 1/20 0.32
CHUK O15111 1/20 0.32
AKT2 P31751 1/20 0.31
MAPT P10636 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA1 Q13131 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5369828 0.76 NPY5R (0.43) ARNPY5RPRKDCMAPTPRKAG1
SCHEMBL5371947 0.74 TYMP (0.38) NPY5RCHRM3
SCHEMBL5371649 0.73 TYMP (0.40) NPY5RCHRM3PDE4APDE4BPDE4C
SCHEMBL5374177 0.70 LMNA (0.43) ARNPY5RSMOCNR2PRKDC
SCHEMBL5372957 0.69 PDE10A (0.34) ARSMOCHRM3PDE4APDE4B
SCHEMBL27379669 0.69 METAP2 (0.37) ARMETAP2SLC6A3GABRA1SMO
SCHEMBL5371106 0.67 KMT2A (0.35) ARSMOCNR2
SCHEMBL5371099 0.67 RAD52 (0.36) RAD52METAP2SLC6A3GABRA1SMO
SCHEMBL5372959 0.66 CNR2 (0.37) ARCHRM3PDE4APDE4BPDE4C
SCHEMBL31539442 0.65 HRH4 (0.45) ARMETAP2SMOPRKDCMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7238212-B2 Imidazole compounds and use of these compounds for dyeing keratinous fibers L'OREAL, S.A. (FR) 2007-07-03 US claimed
US-20050011019-A1 Novel imidazole compounds and use of these compounds for dyeing keratinous fibers L'OREAL, S.A. (FR) 2005-01-20 US claimed
EP-1484049-A1 Imidazole compounds and their use for dyeing of keratinous fibres L'OREAL (FR) 2004-12-08 EP claimed
US-7238212-B2 Imidazole compounds and use of these compounds for dyeing keratinous fibers L'OREAL, S.A. (FR) 2007-07-03 US disclosed
US-20050011019-A1 Novel imidazole compounds and use of these compounds for dyeing keratinous fibers L'OREAL, S.A. (FR) 2005-01-20 US disclosed
EP-1484049-A1 Imidazole compounds and their use for dyeing of keratinous fibres L'OREAL (FR) 2004-12-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050011019-A1 Novel imidazole compounds and use of these compounds for dyeing keratinous fibers KRT18, VIM, NDUFS6 AR 2667/4885NPY5R 3942/4885SLC34A1 3975/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.