SCHEMBL5380413

SCHEMBL5380413

O=c1cc(-c2ccncc2)[nH]c(-c2ccc([N+](=O)[O-])cc2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.56
PKN1 Q16512 2/20 0.56
PKN2 Q16513 2/20 0.56
MAPT P10636 4/20 0.54
MAPK14 Q16539 3/20 0.54
RAB9A P51151 3/20 0.54
CDC7 O00311 2/20 0.54
ALOX5 P09917 2/20 0.54
MEN1 O00255 1/20 0.54
MAPK13 O15264 1/20 0.54
RIPK2 O43353 1/20 0.54
GMNN O75496 1/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.54
CYP3A4 P08684 1/20 0.54
THRB P10828 1/20 0.54
ALOX15 P16050 1/20 0.54
NFKB1 P19838 1/20 0.54
MAPK1 P28482 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377577 0.85 CDC7 (0.49) NPC1PKN1PKN2MAPTRAB9A
SCHEMBL5384093 0.80 GCGR (0.56) NPC1MAPK14RAB9AMAPK13ALDH1A1
SCHEMBL7395689 0.80 MAPK14 (0.48) NPC1MAPTMAPK14RAB9ACDC7
SCHEMBL5399995 0.80 MAPK14 (0.54) MAPK14CDC7ALOX5MAPK13MAPK12
SCHEMBL5380873 0.80 MAPK14 (0.49) MAPTMAPK14CDC7ALOX5MAPK13
SCHEMBL5381545 0.80 CDC7 (0.59) PKN1PKN2MAPTMAPK14CDC7
SCHEMBL5380418 0.78 GSK3B (0.66) NPC1PKN1PKN2MAPTMAPK14
SCHEMBL5383543 0.77 PKN1 (0.53) PKN1PKN2MAPK14CDC7ALOX5
SCHEMBL7133332 0.76 CYP19A1 (0.74) NPC1PKN1PKN2MAPTMAPK14
SCHEMBL3447074 0.74 MAPT (0.62) NPC1PKN1PKN2MAPTMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed