SCHEMBL5382541

SCHEMBL5382541

CN(C)c1nc(-c2cccnc2)cc(=O)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.54
CYP19A1 P11511 1/20 0.47
GSK3B P49841 3/20 0.44
ALK Q9UM73 1/20 0.44
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NPC1 O15118 1/20 0.43
GFER P55789 1/20 0.43
CYP2A6 P11509 2/20 0.43
PKN2 Q16513 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
XDH P47989 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
BTK Q06187 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5384159 0.83 GSK3B (0.64) GSK3BXDHSMN1; SMN2
SCHEMBL5400045 0.80 GSK3B (0.69) KMT2ACYP19A1GSK3BALKALDH1A1
SCHEMBL5382536 0.78 CYP19A1 (0.52) KMT2ACYP19A1ALKALDH1A1CYP2A6
SCHEMBL5384455 0.76 GSK3B (0.75) KMT2ACYP19A1GSK3BALDH1A1HPGD
SCHEMBL14935666 0.75 GSK3B (0.73) KMT2ACYP19A1GSK3BALDH1A1HPGD
SCHEMBL5381426 0.75 GSK3B (0.78) KMT2ACYP19A1GSK3BALDH1A1HPGD
SCHEMBL10840151 0.73 XDH (0.52) KMT2ACYP19A1GSK3BALDH1A1HPGD
SCHEMBL5376063 0.73 GSK3B (0.76) KMT2ACYP19A1GSK3BALDH1A1HPGD
SCHEMBL14935661 0.72 GSK3B (0.55) KMT2AGSK3BPOLBPTGES
SCHEMBL2239607 0.71 CYP2A6 (0.59) KMT2ACYP19A1GSK3BALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed