SCHEMBL5385642

SCHEMBL5385642

O=C(Nc1nc(=O)cc(-c2ccncc2)[nH]1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.51
TTK P33981 1/20 0.51
ITK Q08881 1/20 0.51
AURKB Q96GD4 1/20 0.51
INCENP Q9NQS7 1/20 0.51
F2 P00734 1/20 0.50
F12 P00748 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
MAOB P27338 2/20 0.49
ADORA2A P29274 2/20 0.49
PKM P14618 1/20 0.49
JAK2 O60674 1/20 0.49
TYK2 P29597 1/20 0.49
BACE1 P56817 1/20 0.48
KCNK3 O14649 1/20 0.48
HDAC2 Q92769 1/20 0.47
TBK1 Q9UHD2 1/20 0.46
CDC7 O00311 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5385645 0.80 GSK3B (0.56) AURKATTKITKAURKBINCENP
SCHEMBL3827756 0.79 PIK3C3 (0.53) SMN1; SMN2ADORA2ACDC7MEN1KMT2A
SCHEMBL3827923 0.78 AKR1C3 (0.54) NPC1RAB9AHTTKDM4EL3MBTL1
SCHEMBL24605581 0.76 HDAC6 (0.52) AURKATTKITKAURKBINCENP
SCHEMBL30880097 0.76 HDAC6 (0.52) AURKATTKITKAURKBINCENP
SCHEMBL5380552 0.75 XDH (0.53) SMN1; SMN2RAB9APKMCDC7HTT
SCHEMBL10840691 0.75 CDC7 (0.44) NPC1CDC7
SCHEMBL3825068 0.74 PIK3C3 (0.44) NPC1CDC7
SCHEMBL24867395 0.73 F2 (0.58) AURKATTKITKAURKBINCENP
SCHEMBL5632242 0.72 BUB1 (0.49) SMN1; SMN2HTTKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256199-B1 Pyrimidone derivatives MITSUBISHI CHEMICAL CORPORATION (JP) 2007-08-14 US disclosed
EP-1115721-B1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEM CORP (JP) 2003-12-10 EP disclosed
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed