SCHEMBL539326

SCHEMBL539326

O=C(O)C=CC1CCN(S(=O)(=O)c2ccc(OC(F)(F)F)cc2)C(I)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.42
LIPE Q05469 1/20 0.42
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
EPHX1 P07099 2/20 0.39
MMP9 P14780 2/20 0.39
MMP1 P03956 1/20 0.39
MMP13 P45452 1/20 0.39
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
AKR1C3 P42330 1/20 0.38
HTR2A P28223 1/20 0.38
HSD11B1 P28845 1/20 0.38
TRPA1 O75762 1/20 0.37
DPP4 P27487 3/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424846 0.83 EPHX2 (0.56) EPHX2LIPEKMT2AMEN1EPHX1
SCHEMBL424845 0.83 EPHX2 (0.56) EPHX2LIPEKMT2AMEN1EPHX1
SCHEMBL538758 0.79 EPHX2 (0.46) EPHX2LIPEEPHX1MMP9MMP1
SCHEMBL539061 0.79 EPHX2 (0.46) EPHX2LIPEKMT2AMEN1EPHX1
SCHEMBL2171738 0.76 EPHX2 (0.43) EPHX2LIPEKMT2AMEN1EPHX1
SCHEMBL3717658 0.71 ALDH1A1 (0.56) EPHX2LIPEKMT2AMEN1MMP9
SCHEMBL421549 0.70 EPHX2 (0.62) EPHX2LIPEKMT2AMEN1EPHX1
SCHEMBL421550 0.70 EPHX2 (0.62) EPHX2LIPEKMT2AMEN1EPHX1
SCHEMBL2171525 0.69 MEN1 (0.45) EPHX2LIPEKMT2AMEN1EPHX1
SCHEMBL421636 0.68 EPHX2 (0.57) EPHX2LIPEKMT2AMEN1EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414332-A1 ACRYLAMIDE COMPOUNDS AND THE USE THEREOF Shionogi & Co., Ltd. (JP) 2012-02-08 EP disclosed
WO-2010114181-A1 ACRYLAMIDE COMPOUNDS AND THE USE THEREOF SHIONOGI & CO., LTD. (JP) 2010-10-07 WO disclosed