SCHEMBL5397908

SCHEMBL5397908

CCc1nnc(NS(=O)(=O)c2cccc(Cl)c2C)s1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.59
AKT1 P31749 3/20 0.53
PKM P14618 2/20 0.53
HSD11B1 P28845 4/20 0.51
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
KLKB1 P03952 1/20 0.50
CTSB P07858 1/20 0.50
ELANE P08246 1/20 0.50
HSD17B1 P14061 1/20 0.50
HSD17B2 P37059 1/20 0.50
POLB P06746 3/20 0.49
GAA P10253 1/20 0.49
GPR55 Q9Y2T6 1/20 0.49
EDNRB P24530 1/20 0.49
EDNRA P25101 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA4 P22748 1/20 0.49
CA5A P35218 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5831102 0.88 HSD11B1 (0.49) ATMPKMHSD11B1HSD17B1HSD17B2
SCHEMBL5831070 0.87 HSD11B1 (0.48) ATMHSD11B1HSD17B1HSD17B2EDNRB
SCHEMBL5831386 0.86 HSD11B1 (0.50) ATMPKMHSD11B1HSD17B1HSD17B2
SCHEMBL5830954 0.86 HSD11B1 (0.52) ATMAKT1HSD11B1HSD17B1HSD17B2
SCHEMBL5397833 0.85 HTT (0.52) ATMPKMHSD11B1MEN1KMT2A
SCHEMBL5831865 0.85 ALDH1A1 (0.47) PKMHSD11B1HSD17B1HSD17B2EDNRB
SCHEMBL5831177 0.85 HSD11B1 (0.51) ATMHSD11B1MEN1KMT2AKLKB1
SCHEMBL5831913 0.84 HSD11B1 (0.51) ATMAKT1HSD11B1MEN1KMT2A
SCHEMBL5831410 0.84 HSD11B1 (0.51) ATMAKT1HSD11B1MEN1KMT2A
SCHEMBL5831893 0.84 HSD11B1 (0.46) ATMAKT1HSD11B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070066614-A1 Ihibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2007-03-22 US claimed
US-7173030-B2 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2007-02-06 US claimed
EP-1631558-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2006-03-08 EP claimed
US-20050009821-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2005-01-13 US claimed
WO-2004103980-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2004-12-02 WO claimed
US-20070066614-A1 Ihibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2007-03-22 US disclosed
US-7173030-B2 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB (SE) 2007-02-06 US disclosed
EP-1631558-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2006-03-08 EP disclosed
US-20050009821-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 BIOVITRUM AB 2005-01-13 US disclosed
WO-2004103980-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE I BIOVITRUM AB (SE) 2004-12-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050009821-A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 HSD11B1, HSD17B1, HSD11B2 ATM 4425/4885AKT1 1162/4885PKM 1954/4885
US-20070066614-A1 Ihibitors of 11-beta-hydroxy steroid dehydrogenase type 1 HSD11B1, HSD17B1, HSD17B11 ATM 4338/4885AKT1 2088/4885PKM 2745/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.