SCHEMBL5398290

SCHEMBL5398290

O=C1NC(=O)C2=C1CCN2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 2/20 0.41
PRKD3 O94806 2/20 0.40
PRKCG P05129 2/20 0.40
PRKCB P05771 2/20 0.40
PRKCA P17252 2/20 0.40
PRKCH P24723 2/20 0.40
PRKCI P41743 2/20 0.40
PRKCE Q02156 2/20 0.40
PRKCQ Q04759 2/20 0.40
PRKCZ Q05513 2/20 0.40
PRKCD Q05655 2/20 0.40
PRKD1 Q15139 2/20 0.40
USP7 Q93009 1/20 0.40
USP21 Q9UK80 1/20 0.40
CDK5 Q00535 2/20 0.37
CDK5R1 Q15078 2/20 0.37
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CSNK1A1 P48729 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL710762 0.68
SCHEMBL171230 0.64 CRBN (0.40) CRBNPARP1
SCHEMBL13665462 0.64 CRBN (0.47) CRBNPARP1
SCHEMBL14489609 0.63 CRBN (0.39) CRBNPRKD3PRKCGPRKCBPRKCA
SCHEMBL708902 0.62
SCHEMBL2762093 0.61 ALDH1A1 (0.42) CRBNPARP1
SCHEMBL502060 0.61 ALDH1A1 (0.42) CRBNPARP1
SCHEMBL42430 0.61
SCHEMBL30253370 0.60 CRBN (0.41) CRBNPRKD3PRKCGPRKCBPRKCA
SCHEMBL11133985 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7192967-B1 Cyclic imide-substituted pyridylalkane, alkene, alkine carboxamides useful as cytostatic and immunosuppressive agents ASTELLAS PHARMA GMBH (DE) 2007-03-20 US disclosed
EP-1042315-B1 CYCLIC IMIDE-SUBSTITUTED PYRIDYLALKANE, ALKENE, AND ALKINE CARBOXAMIDES USEFUL AS CYTOSTATIC AND IMMUNOSUPPRESSIVE AGENTS KLINGE CO CHEM PHARM FAB (DE) 2004-04-14 EP disclosed