SCHEMBL5400840

SCHEMBL5400840

CC(CCc1ccccc1F)(c1ccccc1F)C1(O)CCN(Cc2ccc[nH]c2=O)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.37
CCR8 P51685 1/20 0.37
ALDH1A1 P00352 6/20 0.36
KDM4E B2RXH2 5/20 0.36
POLB P06746 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
MAPK1 P28482 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
CYP2A13 Q16696 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
OPRM1 P35372 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1474804 0.79 ALDH1A1 (0.41) KCNH2CCR8ALDH1A1KDM4EPOLB
SCHEMBL12827514 0.74 ALDH1A1 (0.48) KCNH2CCR8ALDH1A1CYP1A2CYP3A4
SCHEMBL5400844 0.74 DPP4 (0.38) KCNH2CCR8ALDH1A1KDM4EPOLB
SCHEMBL5400852 0.72 USP7 (0.37) KCNH2CCR8ALDH1A1KDM4EPOLB
SCHEMBL5400845 0.71 TACR1 (0.42) KCNH2CCR8ALDH1A1KMT2AMEN1
SCHEMBL1476057 0.70 CCR8 (0.38) KCNH2CCR8ALDH1A1KDM4EPOLB
SCHEMBL1476956 0.70 KCNH2 (0.44) KCNH2CCR8ALDH1A1KDM4EPOLB
SCHEMBL1476401 0.69 TACR2 (0.46) KCNH2ALDH1A1KDM4EPOLBCYP1A2
SCHEMBL1475562 0.69 KCNH2 (0.40) KCNH2CCR8ALDH1A1KDM4EPOLB
SCHEMBL1474461 0.69 KCNH2 (0.40) KCNH2CCR8ALDH1A1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7265108-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI CO., LTD. (JP) 2007-09-04 US disclosed