SCHEMBL5400845

SCHEMBL5400845

O=c1[nH]cccc1CN1CCC(O)(CC(CCc2ccccc2F)c2ccc(F)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.42
USP7 Q93009 3/20 0.40
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
CCR8 P51685 1/20 0.37
KCNH2 Q12809 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
GAA P10253 1/20 0.34
ALDH1A1 P00352 2/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5400852 0.90 USP7 (0.37) TACR1USP7DRD2DRD4DRD3
SCHEMBL1474804 0.82 ALDH1A1 (0.41) USP7DRD2DRD4DRD3CCR8
SCHEMBL5400844 0.79 DPP4 (0.38) TACR1USP7DRD2DRD4DRD3
SCHEMBL1476956 0.75 KCNH2 (0.44) USP7DRD2DRD4DRD3CCR8
SCHEMBL12827514 0.73 ALDH1A1 (0.48) DRD2DRD4DRD3CCR8KCNH2
SCHEMBL5400840 0.71 KCNH2 (0.37) CCR8KCNH2MEN1KMT2AGAA
SCHEMBL1475562 0.70 KCNH2 (0.40) CCR8KCNH2KMT2AGAAALDH1A1
SCHEMBL1475951 0.70 CCR8 (0.42) CCR8KCNH2MEN1KMT2AATM
SCHEMBL1476057 0.69 CCR8 (0.38) USP7DRD2DRD4DRD3CCR8
SCHEMBL1475312 0.68 KCNH2 (0.43) CCR8KCNH2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7265108-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI CO., LTD. (JP) 2007-09-04 US disclosed