SCHEMBL5400852

SCHEMBL5400852

O=c1[nH]cccc1CN1CCC(O)(CC(CCc2ccccc2F)c2ccccc2F)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP7 Q93009 1/20 0.37
CCR8 P51685 1/20 0.35
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 4/20 0.34
KMT2A Q03164 3/20 0.34
TACR1 P25103 2/20 0.34
MEN1 O00255 2/20 0.34
ATM Q13315 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
MCHR1 Q99705 1/20 0.34
KDM4E B2RXH2 3/20 0.33
CYP2A13 Q16696 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5400845 0.90 TACR1 (0.42) USP7CCR8KCNH2ALDH1A1KMT2A
SCHEMBL1474804 0.83 ALDH1A1 (0.41) USP7CCR8KCNH2ALDH1A1KMT2A
SCHEMBL5400844 0.80 DPP4 (0.38) USP7CCR8KCNH2ALDH1A1KMT2A
SCHEMBL12827514 0.74 ALDH1A1 (0.48) CCR8KCNH2ALDH1A1KMT2AMEN1
SCHEMBL1476956 0.74 KCNH2 (0.44) USP7CCR8KCNH2ALDH1A1KMT2A
SCHEMBL5400840 0.72 KCNH2 (0.37) CCR8KCNH2ALDH1A1KMT2AMEN1
SCHEMBL1475951 0.70 CCR8 (0.42) CCR8KCNH2ALDH1A1KMT2AMEN1
SCHEMBL1476057 0.70 CCR8 (0.38) USP7CCR8KCNH2ALDH1A1KMT2A
SCHEMBL1475562 0.69 KCNH2 (0.40) CCR8KCNH2ALDH1A1KMT2AKDM4E
SCHEMBL1475313 0.69 MCHR1 (0.39) USP7ALDH1A1MCHR1KDM4EOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7265108-B2 Nitrogen containing heterocyclic compounds and medicines containing the same EISAI CO., LTD. (JP) 2007-09-04 US disclosed