SCHEMBL5402329

SCHEMBL5402329

COc1ccc(CN(CCC(=O)O)C(=O)c2ccccc2-c2ccccc2C(=O)NCc2cccc(C)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.55
HDAC1 Q13547 4/20 0.52
HDAC6 Q9UBN7 4/20 0.52
TDP1 Q9NUW8 1/20 0.48
NPC1 O15118 1/20 0.47
TSHR P16473 2/20 0.47
HPGD P15428 3/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 1/20 0.47
LPAR1 Q92633 5/20 0.47
USP2 O75604 1/20 0.45
APEX1 P27695 1/20 0.44
PDK1 Q15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5392918 0.93 RAB9A (0.65) RAB9AHDAC1HDAC6TDP1TSHR
SCHEMBL4928557 0.93 KDM4E (0.54) RAB9AHDAC1HDAC6TDP1TSHR
SCHEMBL5409793 0.92 RAB9A (0.54) RAB9AHDAC1HDAC6NPC1HPGD
SCHEMBL5397479 0.92 HDAC1 (0.61) RAB9AHDAC1HDAC6TDP1NPC1
SCHEMBL5407093 0.92 HDAC1 (0.61) RAB9AHDAC1HDAC6TDP1NPC1
SCHEMBL5392370 0.91 HDAC1 (0.55) RAB9AHDAC1HDAC6TDP1NPC1
SCHEMBL5403175 0.91 HDAC1 (0.59) RAB9AHDAC1HDAC6TDP1NPC1
SCHEMBL5406209 0.90 RAB9A (0.54) RAB9AHDAC1HDAC6TDP1TSHR
SCHEMBL5409746 0.90 RAB9A (0.54) RAB9AHDAC1HDAC6TDP1NPC1
SCHEMBL5397034 0.90 RAB9A (0.69) RAB9AHDAC1HDAC6TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285680-B2 β-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-10-23 US disclosed
US-20050256160-A1 Beta-alanine derivatives and the use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2005-11-17 US disclosed
EP-1533294-A1 BETA-ALANINE DERIVATIVE AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256160-A1 Beta-alanine derivatives and the use thereof TGFB1, PML, APOB RAB9A 3132/4885HDAC1 2189/4885HDAC6 2386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.