SCHEMBL5406664

SCHEMBL5406664

CCCCn1nc(-c2ccccc2)c2ccc(C(F)(F)F)cc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 2/20 0.53
ESR1 P03372 2/20 0.47
KDM4E B2RXH2 2/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CYP1A2 P05177 3/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
KIF11 P52732 1/20 0.44
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
CRHBP P24387 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5409012 0.90 KDM4E (0.46) PTGER1ESR1KDM4ETSHRHSD17B10
SCHEMBL4030236 0.88 ESR1 (0.57) PTGER1ESR1KDM4ECYP1A2CYP2C9
SCHEMBL4029629 0.84 ESR1 (0.52) PTGER1ESR1KDM4ECYP1A2CYP2C9
SCHEMBL5418980 0.80 ALDH1A1 (0.63) PTGER1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL4029018 0.79 ESR1 (0.51) PTGER1ESR1KDM4ETSHRHSD17B10
SCHEMBL15631875 0.77 LMNA (0.69) PTGER1KDM4ETSHRHSD17B10CYP1A2
SCHEMBL4035483 0.74 ESR1 (0.44) PTGER1ESR1KDM4ECYP2C9CYP2C19
SCHEMBL4035081 0.74 ESR1 (0.57) PTGER1ESR1CYP1A2CYP2C9CYP2C19
SCHEMBL4028897 0.74 ESR1 (0.61) PTGER1ESR1CYP1A2CYP2C9CYP2C19
SCHEMBL594869 0.73 CNR2 (0.52) ALDH1A1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7241791-B2 Substituted 4-(indazol-3-yl)phenols WYETH (US) 2007-07-10 US disclosed